YOSHIDA Masahito
- Articles
- Conformation-based Design and Synthesis of Apratoxin A Mimetics Modified at the alfa,beta-Unsaturated Thiazoline Moiety
Onda Yuichi; Masuda Yuichi; Yoshida Masahito; Doi Takayuki
J. Med. Chem./60(15)/pp.6751-6765, 2017-08 - Facile Synthesis of Pyrrolyl 4-Quinolinone Alkaloids Quinolactacide by 9-AJ Catalyzed Tandem Acyl Transfer-Cyclization of o-Alkynoylaniline Derivatives
Yoshida Masahito; Saito Koya; Uekusa Hidehiro; Doi Takayuki
ACS Omega/2(8)/pp.4370-4381, 2017-08 - Stereoselective Synthesis of beta-Amino Acid Derivatives by Asymmetric Mannich Reaction in Flow
Yoshida Masahito; Umeda Koji; Doi Takayuki
Bull. Chem. Soc. Jpn./90(10)/pp.1157-1163, 2017-07 - Potent oxazoline analog of apratoxin C: Synthesis, biological evaluation, and conformational analysis
Yoshida Masahito; Onda Yuichi; Masuda Yuichi; Doi Takayuki
Biopolymers (Pept. Sci.)/106(4)/pp.404-14, 2016-11 - Combinatorial Solid-Phase Synthesis and Biological Evaluation of Cyclodepsipeptide Destruxin B as a Negative regulator for Osteoclast Morphology
Sato Hiroshi; Yoshida Masahito; Murase Hayato; Nakagawa ...
ACS Combi. Sci./18(9)/pp.590-595, 2016-09 - Design, Synthesis, and Biological Evaluation of Beauveriolide Analogues Bearing Photoreactive Amino Acids
Masuda Yuichi; Aoyama Kazumasa; Yoshida Masahito; Kobayas...
Chem. Pharm. Bull./64(7)/pp.754-765, 2016-07 - Solid-Phase Combinatorial Synthesis and Biological Evaluation of Destruxin E Analogues
Yoshida Masahito; Ishida Yoshitaka; Adachi Kenta; Murase ...
Chem. Eur. J./21(50)/pp.18417-18430, 2015-12 - Total Synthesis Cyclodepsipeptide Spiruchostatin A on Silyl-linker polymer-support
Yoshida Masahito; Sasahara Ken-ichi; Doi Takayuki
Tetrahdron/71(40)/pp.7647-7653, 2015-08 - Pyrrolidine-containing peptides, JBIR-126, -148, and -149, from Streptomyces sp. NBRC 111228
Izumikawa Miho; Kawahara Teppei; Kagaya Noritaka; Yamamur...
Tetrahedron Lett./56(39)/pp.5333-5336, 2015-08 - Study for diastereoselective aldol reaction in flow: synthesis of (E)-(S)-3-hydroxy-7-tritylthio-4-heptenoic acid, a key component of cyclodepsipeptide HDAC inhibitors
Doi Takayuki; Otaka Hiroyuki; Umeda Koji; Yoshida Masahito
Tetradedron/71(37)/pp.6463-6470, 2015-05 - Synthesis and biological evaluation of c-aromataxane derivatives as p-glycoprotein-mediated multi drug resistance reversal agents
Doi Takayuki; Yamaguchi Naoko; Ohsawa Kosuke; Nakai Kazu...
Heterocycles/90(1)/pp.482-501, 2015-01 - Total Synthesis and Structure Elucidation of JBIR‐39: A Linear Hexapeptide Possessing Piperazic Acid and γ‐Hydroxypiperazic Acid Residues
Yoshida Masahito; Sekioka Naoki; Izumikawa Miho; Kozone ...
Chem. Eur. J./21(7)/pp.3031-3041, 2014-12 - An Efficient Synthesis of Aurone Derivatives by the Tributylphosphine-catalyzed Regioselective Cyclization of o-Alkynoylphenols
Saito Koya; Yoshida Masahito; Doi Takayuki
Chem. Lett./44(2)/pp.141-143, 2014-11 - An Efficient Partial Reduction of α,β-Unsaturated Esters Using DIBAL-H in FLow
Yoshida Masahito; Otaka Hiroyuki; Doi Takayuki
European Journal of Organic Chemistry/27/pp.6010-6016, 2014-09 - Total Synthesis and Conformational Analysis of Apratoxin C
Masuda Yuichi; Suzuki Jun; Onda Yuichi; Fujino Yuta; ...
The Journal of Organic Chemistry/79(17)/pp.8000-8009, 2014-09 - A Concise Total Synthesis of Biologically Active Frutinones via Tributylphosphine-catalyzed Tandem Acyl Transfer-Cyclization
Yoshida Masahito; Saito Koya; Fujino Yuta; Doi Takayuki
Tetrahedron/70(21)/pp.3452-3458, 2014-05 - Epigallocatechin gallate decreases the micellar solubility of cholesterol via specific interaction with phosphatidylcholine
Kobayashi Makoto; Nishizawa Masato; Inoue Nao; Hosoya ...
Journal of Agricultural and Food Chemistry/62(13)/pp.2881-2890, 2014-04 - Scalable Solution-Phase Synthesis of the Biologically Active Cyclodepsipeptide Destruxin E, a Potent Negative Regulator of Osteoclast Morphology
Yoshida Masahito; Sato Hiroshi; Ishida Yoshitaka; Naka...
The Journal of Organic Chemistry/79(1)/pp.296-306, 2014-01 - Total Synthesis and Characterization of Thielocin B1 as a Protein－Protein Interaction Inhibitor of PAC3 Homodimer
Doi Takayuki; Yoshida Masahito; Ohsawa Kosuke; Shin-ya K...
Chemical Science/5/pp.1860-1868, 2014-01 - Synthesis of Hepta-oxazole Macrocyclic Analogues of Telomestatin and Evaluation of Their Telomerase Inhibitory Activities,
Shibata Kazuaki; Yoshida Masahito; Takahashi Takashi; Tak...
Bulletin of Chemical Society of Japan/86(12)/pp.1453-1465, 2013-08 - A Direct and Mild Formylation Method for Substituted Benzenes Utilizing Dichloromethyl Methyl Ether-Silver Trifluoromethanesulfonate
Ohsawa Kosuke; Yoshida Masahito; Doi Takayuki
The Journal of Organic Chemistry/78(7)/pp.3438-3444, 2013-04 - A Concise Synthesis of 3-Aroylflavones via Lewis Base 9-Azajulolidine－catalyzed Tandem Acyl Transfer－Cyclization
Yoshida Masahito; Saito Koya; Fujino Yuta; Doi Takayuki
Chemical Communications/48/pp.11796-11798, 2012-10 - Development of a Near Infrared Fluorescence Labeling Reagent: Synthesis of Indole-Functionalized Indocyanine Green Derivatives
Doi Takayuki; Oikawa Koya; Suzuki Jun; Yoshida Masahito; ...
Synlett/(2)/pp.306-310, 2012-02 - Conformationally Restricted Analog and Biotin-Labeled Probe Based on Beauveriolide III
Doi Takayuki; Muraoka Terushige; Ohshiro Taichi; Matsu...
Bioorganic & medicinal chemistry letters/22(1)/pp.696-699, 2012-01 - Regioselective Synthesis of Flavone Derivatives via DMAP-catalyzed Cyclization of o-Alkynoylphenols
Yoshida Masahito; Fujino Yuta; Saito Koya; Doi Takayuki
Tetrahedron/67(51)/pp.9993-9997, 2011-12 - more...
- Conformation-based Design and Synthesis of Apratoxin A Mimetics Modified at the alfa,beta-Unsaturated Thiazoline Moiety